Basic Peptide Information

DICL ID
DICL_Pep_00657
Ion Channel
Voltage-gated sodium channel type 2 subunit alpha
Peptide Function
Inhibitor
Gene Name
SCN2A

Activity Data (nM)

IC50
130 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
DCLGWFKSCDPKNDKCCKNYSCSRRDRWCKYDL
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
β-TrtX-Cd1a
Peptide Species
Ceratogyrus darlingi (Rear horned baboon tarantula)
Peptide Name
Beta-theraphotoxin-Cd1a
CAS Number
Not available

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−100 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
HEK293 cell (Homo sapiens embryonic kidney 293 cell)

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available